Infliximab levels predict ASUC outcomes

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Early infliximab drug monitoring may predict short-term outcomes and identify acute severe ulcerative colitis (ASUC) patients who could benefit from intensified dosing, according to data from the multicenter PREDICT-UC study.

The goal of the PREDICT‑UC trial was to determine whether intensified or accelerated infliximab induction regimens are superior to standard infliximab induction for treating steroid‑refractory ASUC and to explore how infliximab drug levels and clearance relate to treatment response.

In a prospective observational study published in Gastroenterology, Australian researchers measured serum and fecal infliximab levels and modeled drug clearance during the first weeks of rescue therapy in 135 patients with steroid-refractory ASUC enrolled in PREDICT-UC. Nearly two-thirds of patients (63%) responded by day 7, but 27% experienced treatment failure by day 14 and 13% required colectomy within 3 months.

A key finding was the prognostic value of early serum infliximab exposure. Lower day 3 serum infliximab levels were associated with both day 14 treatment failure and subsequent colectomy. A day 3 level of 57.9 µg/mL or less identified patients at high risk for colectomy with 83.3% sensitivity, 67% specificity, and a negative predictive value of nearly 97%, suggesting early reassurance may be possible when levels are adequate, noted Christopher F.D. Li Wai Suen, MD, of the University of Melbourne, Department of Medicine, Australia, and colleagues.

Infliximab clearance emerged as another important determinant of outcome. Higher early clearance, especially by day 7, was strongly associated with nonresponse, treatment failure, and colectomy. Notably, patients with high clearance were more likely to respond to an initial 10 mg/kg dose than to standard 5 mg/kg dosing, and intensified induction appeared to mitigate colectomy risk in this subgroup.

Fecal infliximab levels correlated with inflammatory burden and endoscopic severity, supporting the concept of luminal drug loss in severe disease. Although management was not adjusted based on drug levels, the findings provide a rationale for early infliximab monitoring in ASUC.

“This study supports observational data indicating infliximab clearance to be a major determinant of outcomes in ASUC, and for the first time demonstrates that increased clearance may potentially be overcome by more intensive dosing,” the authors wrote.

Biological specimens for the current study were derived from a clinical trial that was supported by a Janssen-Cilag investigator-initiated study grant. Many of the authors reported financial relationships with pharmaceutical companies, including speaker/consulting fees and research funding.

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